Influence of CYP2D6 ,CYP3A4 ,CYP3A5 and ABCB1 Polymorphisms on Pharmacokinetics and Safety of Aripiprazole in Healthy Volunteers

Author:

Belmonte Carmen12,Ochoa Dolores12,Román Manuel12,Saiz-Rodríguez Miriam1,Wojnicz Aneta1,Gómez-Sánchez Clara Isabel3,Martín-Vílchez Samuel1,Abad-Santos Francisco124

Affiliation:

1. Clinical Pharmacology Department; Hospital Universitario de la Princesa; Instituto Teofilo Hernando; Instituto de Investigacion Sanitaria Princesa (IP); Madrid Spain

2. UICEC Hospital Universitario de la Princesa, Plataforma SCReN (Spanish Clinical Reseach Network); Instituto de Investigacion Sanitaria la Princesa (IP); Madrid Spain

3. Department of Genetics; IIS-Fundacion Jimenez Dıaz University Hospital (IIS-FJD, UAM); Madrid Spain

4. Center for Biomedical Research Network Hepatic and Liver diseases (CIBERedh) - Instituto de Salud Carlos III; Madrid Spain

Publisher

Wiley

Subject

Pharmacology,Toxicology,General Medicine

Reference52 articles.

1. Food and Drug Administration Aripiprazole label 2014 http://www.accessdata.fda.gov/drugsatfda_docs/label/2014/021436s038,021713s030,021729s022,021866s023lbl.pdf

2. Aripiprazole, a novel antipsychotic, is a high-affinity partial agonist at human dopamine D2 receptors;Burris;J Pharmacol Exp Ther,2002

3. The antipsychotic aripiprazole is a potent, partial agonist at the human 5-HT1A receptor;Jordan;Eur J Pharmacol,2002

4. Aripiprazole, a novel atypical antipsychotic drug with a unique and robust pharmacology;Shapiro;Neuropsychopharmacology,2003

5. Aripiprazole: profile on efficacy and safety;Goodnick;Expert Opin Pharmacother,2002

同舟云学术

1.学者识别学者识别

2.学术分析学术分析

3.人才评估人才评估

"同舟云学术"是以全球学者为主线,采集、加工和组织学术论文而形成的新型学术文献查询和分析系统,可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容,当前同舟云学术共收录了国内外主流学术期刊6万余种,收集的期刊论文及会议论文总量共计约1.5亿篇,并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询!咨询电话:010-8811{复制后删除}0370

www.globalauthorid.com

TOP

Copyright © 2019-2024 北京同舟云网络信息技术有限公司
京公网安备11010802033243号  京ICP备18003416号-3