N‐lockingstabilization of covalent helical peptides: Application to Bfl‐1 antagonists-Reference-Cited by-同舟云学术

N‐lockingstabilization of covalent helical peptides: Application to Bfl‐1 antagonists

Published:2020-04 Issue:4 Volume:95 Page:412-426
ISSN:1747-0277
Container-title:Chemical Biology & Drug Design
language:en
Short-container-title:Chem Biol Drug Des

Author:

Baggio Carlo¹,Udompholkul Parima¹,Gambini Luca¹,Jossart Jennifer²,Salem Ahmed F.¹,Håkansson Maria³,Perry J. Jefferson P.²^ORCID,Pellecchia Maurizio¹^ORCID

Affiliation:

1. Division of Biomedical Sciences School of Medicine University of California Riverside Riverside CA USA

2. Department of Biochemistry College of Natural and Agricultural Sciences University of California Riverside Riverside CA USA

3. SARomics Biostructures AB Lund Sweden

Funder

National Institutes of Health

Publisher

Wiley

Subject

Molecular Medicine,Biochemistry,Drug Discovery,Pharmacology,Organic Chemistry

Link

https://onlinelibrary.wiley.com/doi/pdf/10.1111/cbdd.13661

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1. An antiapoptotic BCL-2 family expression index predicts the response of chronic lymphocytic leukemia to ABT-737

2. Design of Potent pan-IAP and Lys-Covalent XIAP Selective Inhibitors Using a Thermodynamics Driven Approach

3. Enthalpy-Based Screening of Focused Combinatorial Libraries for the Identification of Potent and Selective Ligands

4. hBfl-1/hNOXA Interaction Studies Provide New Insights on the Role of Bfl-1 in Cancer Cell Resistance and for the Design of Novel Anticancer Agents

5. Downsizing Proto-oncogene cFos to Short Helix-Constrained Peptides That Bind Jun

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