Synthesis and Evaluation of Biological and Antitumor Activities of Tetrahydrobenzothieno[2,3-d]Pyrimidine Derivatives as Novel Inhibitors of FGFR1-Reference-Cited by-同舟云学术

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Synthesis and Evaluation of Biological and Antitumor Activities of Tetrahydrobenzothieno[2,3-d]Pyrimidine Derivatives as Novel Inhibitors of FGFR1

Published:2016-02-01 Issue:4 Volume:87 Page:499-507
ISSN:1747-0277
Container-title:Chemical Biology & Drug Design
language:en
Short-container-title:Chem Biol Drug Des

Author:

Wang Xuebao¹,Chen Di¹,Yu Shufang¹,Zhang Zaikui¹,Wang Yu¹,Qi Xiaolu²,Fu Weitao¹,Xie Zixin¹,Ye Faqing¹

Affiliation:

1. School of Pharmaceutical Sciences; Wenzhou Medical University; Wenzhou 325035 China

2. Yichang Humanwell Pharmaceutical Co., Ltd; Yichang 443005 China

Funder

National Natural Science Foundation of China

Publisher

Wiley

Subject

Molecular Medicine,Biochemistry,Drug Discovery,Pharmacology,Organic Chemistry

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1111/cbdd.12687/fullpdf

Reference28 articles.

1. Fibroblast growth factor signalling: from development to cancer;Turner;Nat Rev Cancer,2010

2. Tyrosine kinases in disease: overview of kinase inhibitors as therapeutic agents and current drugs in clinical trials;Strawn;Expert Opin Investig Drugs,1998

3. Small molecule inhibition of fibroblast growth factor receptors in cancer;Liang;Cytokine Growth Factor Rev,2013

4. FGFR1 mutations in Rosette-forming glioneuronal tumors of the fourth ventricle;Gessi;J Neuropathol Exp Neurol,2014

5. Discovery of 3-(2, 6-dichloro-3, 5-dimethoxy-phenyl)-1-{6-[4-(4-ethyl-piperazin-1-yl) -phenylamino]-pyrimidin-4-yl}-1-methyl-urea (NVP-BGJ398), a potent and selective inhibitor of the fibroblast growth factor receptor family of receptor tyrosine kinase;Guagnano;J Med Chem,2011

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