Estimation of competitive antagonist affinity from functional inhibition curves using the Gaddum, Schild and Cheng-Prusoíf equations
Author:
Publisher
Wiley
Subject
Pharmacology
Link
http://onlinelibrary.wiley.com/wol1/doi/10.1111/j.1476-5381.1993.tb13737.x/fullpdf
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4. Antagonist binding properties of five cloned muscarinic receptors expressed in CHO-K1 cells;BUCKLEY;Mol. Pharmacol.,1989
5. Relationship between the inhibition constant (Ki) and the concentration of an inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction;CHENG;Biochem. Pharmacol.,1973
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