FFA1-selective agonistic activity based on docking simulation using FFA1 and GPR120 homology models-Reference-Cited by-同舟云学术

FFA1-selective agonistic activity based on docking simulation using FFA1 and GPR120 homology models

Published:2013-03-12 Issue:7 Volume:168 Page:1570-1583
ISSN:0007-1188
Container-title:British Journal of Pharmacology
language:en
Short-container-title:Br J Pharmacol

Author:

Takeuchi Masato,Hirasawa Akira,Hara Takafumi,Kimura Ikuo,Hirano Tatsuya,Suzuki Takayoshi,Miyata Naoki,Awaji Takeo,Ishiguro Masaji,Tsujimoto Gozoh

Publisher

Wiley

Subject

Pharmacology

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1111/j.1476-5381.2012.02052.x/fullpdf

Reference32 articles.

1. Akerman M Houze J Lin DCH Liu J Luo J Medina JC et al 2005 Arylmethoxyphenyl-alkylcarboxylic acids and related derivatives for use in treating metabolic disorders

2. Guide to Receptors and Channels (GRAC), 5th Edition;Alexander;Br J Pharmacol,2011

3. Discovery of diacylphloroglucinols as a new class of GPR40 (FFAR1) agonists;Bharate;Bioorg Med Chem Lett,2008

4. The orphan G protein-coupled receptor GPR40 is activated by medium and long chain fatty acids;Briscoe;J Biol Chem,2003

5. Pharmacological regulation of insulin secretion in MIN6 cells through the fatty acid receptor GPR40: identification of agonist and antagonist small molecules;Briscoe;Br J Pharmacol,2006

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