Supra-physiological efficacy at GPCRs: superstition or super agonists?
Author:
Affiliation:
1. Drug Discovery Biology; Monash Institute of Pharmaceutical Sciences; Monash University; Parkville Vic. Australia
Publisher
Wiley
Subject
Pharmacology
Link
http://onlinelibrary.wiley.com/wol1/doi/10.1111/bph.12142/fullpdf
Reference16 articles.
1. Restructuring G-protein-coupled receptor activation;Audet;Cell,2012
2. Operational models of pharmacological agonism;Black;Proc R Soc Lond B Biol Sci,1983
3. Structure of the adenosine A2A receptor in complex with ZM241385 and the xanthines XAC and caffeine;Doré;Structure,2011
4. On the analysis of ligand-directed signaling at G protein-coupled receptors;Ehlert;Naunyn Schmiedebergs Arch Pharmacol,2008
5. The strange case of TGN1412;Farzaneh;Cancer Immunol Immunother,2007
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