Author:
AL-OBEIDI FAHAD,O'CONNOR STEVEN D.,JOB CONSTANTIN,HRUBY VICTOR J.,PETTITT B. MONTGOMERY
Subject
Endocrinology,Biochemistry
Cited by
26 articles.
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1. Discovery of a β-Hairpin Octapeptide, c[Pro-Arg-Phe-Phe-Dap-Ala-Phe-DPro], Mimetic of Agouti-Related Protein(87–132) [AGRP(87–132)] with Equipotent Mouse Melanocortin-4 Receptor (mMC4R) Antagonist Pharmacology;Journal of Medicinal Chemistry;2015-06
2. 1,4-Disubstituted-[1,2,3]triazolyl-Containing Analogues of MT-II: Design, Synthesis, Conformational Analysis, and Biological Activity;Journal of Medicinal Chemistry;2014-11-13
3. Structure–Activity Relationships of Peptides Incorporating a Bioactive Reverse-Turn Heterocycle at the Melanocortin Receptors: Identification of a 5800-fold Mouse Melanocortin-3 Receptor (mMC3R) Selective Antagonist/Partial Agonist versus the Mouse Melanocortin-4 Receptor (mMC4R);Journal of Medicinal Chemistry;2013-03-25
4. Conformational study on cyclic melanocortin ligands and new insight into their binding mode at the MC4 receptor;European Journal of Medicinal Chemistry;2011-09
5. Combinatorial Library Synthesis and Biological Evaluation of Pyrazolo[4,3-e][1,4]diazepine as a Potential Privileged Structure;ChemMedChem;2009-05-11