Covalent modification of GABAAreceptor isoforms by a diazepam analogue provides evidence for a novel benzodiazepine binding site that prevents modulation by these drugs-Reference-Cited by-同舟云学术

Covalent modification of GABAAreceptor isoforms by a diazepam analogue provides evidence for a novel benzodiazepine binding site that prevents modulation by these drugs

Published:2008-09 Issue:6 Volume:106 Page:2353-2363
ISSN:0022-3042
Container-title:Journal of Neurochemistry
language:en
Short-container-title:

Author:

Baur Roland,Tan Kelly R.,Lüscher Benjamin P.,Gonthier Anne,Goeldner Maurice,Sigel Erwin

Publisher

Wiley

Subject

Cellular and Molecular Neuroscience,Biochemistry

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1111/j.1471-4159.2008.05574.x/fullpdf

Reference28 articles.

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3. Towards a relative orientation of benzodiazepines in their binding pocket on GABAA receptors;Berezhnoy;J. Biol. Chem.,2004

4. Conformational changes at benzodiazepine binding sites of GABAA receptors detected with a novel technique;Berezhnoy;J. Neurochem.,2005

5. The relative amount of cRNA coding for γ2 subunits affects stimulation by benzodiazepines in GABAA receptors expressed in Xenopus oocytes;Boileau;Neuropharmacology,2002

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