Replacement of histidine in position 105 in the α5subunit by cysteine stimulates zolpidem sensitivity of α5β2γ2GABAAreceptors
Author:
Publisher
Wiley
Subject
Cellular and Molecular Neuroscience,Biochemistry
Link
http://onlinelibrary.wiley.com/wol1/doi/10.1111/j.1471-4159.2007.04982.x/fullpdf
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3. Zolpidem Activation of Alpha 1-Containing GABAA Receptors Selectively Inhibits High Frequency Action Potential Firing of Cortical Neurons;Frontiers in Pharmacology;2019-01-09
4. International Union of Basic and Clinical Pharmacology. CVI: GABAA Receptor Subtype- and Function-selective Ligands: Key Issues in Translation to Humans;Pharmacological Reviews;2018-10
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