Understanding inhibitor resistance in Mps1 kinase through novel biophysical assays and structures-Reference-Cited by-同舟云学术

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Understanding inhibitor resistance in Mps1 kinase through novel biophysical assays and structures

Published:2017-09 Issue:35 Volume:292 Page:14496-14504
ISSN:0021-9258
Container-title:Journal of Biological Chemistry
language:en
Short-container-title:Journal of Biological Chemistry

Author:

Hiruma Yoshitaka,Koch Andre,Hazraty Nazila,Tsakou Foteini,Medema René H.,Joosten Robbie P.,Perrakis Anastassis

Funder

Nederlandse Organisatie voor Wetenschappelijk Onderzoek

KWF Kankerbestrijding

Publisher

Elsevier BV

Subject

Cell Biology,Molecular Biology,Biochemistry

Reference39 articles.

1. Genetic instability in colorectal cancers;Lengauer;Nature,1997

2. The MPS1 family of protein kinases;Liu;Annu. Rev. Biochem,2012

3. A chemical tool box defines mitotic and interphase roles for Mps1 kinase;Lan;J. Cell Biol,2010

4. Inhibition of the spindle assembly checkpoint kinase TTK enhances the efficacy of docetaxel in a triple-negative breast cancer model;Maia;Ann. Oncol,2015

5. Structure-based design of orally bioavailable 1 H-pyrrolo[3,2-c]pyridine inhibitors of mitotic kinase monopolar spindle 1 (MPS1);Naud;J. Med. Chem,2013

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2. Development of MPS1 Inhibitors: Recent Advances and Perspectives;Journal of Medicinal Chemistry;2023-12-14

3. How Ligands Interact with the Kinase Hinge;ACS Medicinal Chemistry Letters;2023-10-09

4. Augmenting bioactivity by docking‐generated multiple ligand poses to enhance machine learning and pharmacophore modelling: discovery of new TTK inhibitors as case study;Molecular Informatics;2023-06

5. New cyclic glycolipids from Silene succulenta promote in vitro MCF-7 breast carcinoma cell apoptosis by cell cycle arrest and in silico mitotic Mps1/TTK inhibition;RSC Advances;2023

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