Metabolomics and proteomics identify the toxic form and the associated cellular binding targets of the anti-proliferative drug AICAR
Author:
Funder
Ligue contre le Cancer
Publisher
Elsevier BV
Subject
Cell Biology,Molecular Biology,Biochemistry
Reference35 articles.
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2. 5-Aminoimidazole-4-carboxamide-1-β-d-ribofuranosyl 5′-monophosphate (AICAR), a highly conserved purine intermediate with multiple effects;Daignan-Fornier;Metabolites,2012
3. The AMPK agonist AICAR inhibits the growth of EGFRvIII-expressing glioblastomas by inhibiting lipogenesis;Guo;Proc. Natl. Acad. Sci. U.S.A,2009
4. 5-Aminoimidazole-4-carboxamide-1-β-d-ribofuranoside inhibits cancer cell proliferation in vitro and in vivo via AMP-activated protein kinase;Rattan;J. Biol. Chem,2005
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1. Lethal metabolism of Candida albicans respiratory mutants;PLOS ONE;2024-04-05
2. Treatment of AICA ribosiduria by suppression of de novo purine synthesis;Molecular Genetics and Metabolism;2024-03
3. Anti-tumor activity of 5-aminoimidazole-4-carboxamide riboside with AMPK-independent cell death in human adult T-cell leukemia/lymphoma;European Journal of Pharmacology;2023-12
4. An intrinsic purine metabolite AICAR blocks lung tumour growth by targeting oncoprotein mucin 1;British Journal of Cancer;2023-02-21
5. Metabolites of De Novo Purine Synthesis: Metabolic Regulators and Cytotoxic Compounds;Metabolites;2022-12-02
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