The anticancer thiosemicarbazones Dp44mT and triapine lack inhibitory effects as catalytic inhibitors or poisons of DNA topoisomerase IIα-Reference-Cited by-同舟云学术

登录注册会员服务联系我们

The anticancer thiosemicarbazones Dp44mT and triapine lack inhibitory effects as catalytic inhibitors or poisons of DNA topoisomerase IIα

Published:2012-07 Issue:1 Volume:84 Page:52-58
ISSN:0006-2952
Container-title:Biochemical Pharmacology
language:en
Short-container-title:Biochemical Pharmacology

Author:

Yalowich Jack C.,Wu Xing,Zhang Rui,Kanagasabai Ragu,Hornbaker Marisa,Hasinoff Brian B.

Funder

Canadian Institutes of Health Research

Canada Research Chairs Program

Canada Research Chair in Drug Development

NIH

Publisher

Elsevier BV

Subject

Pharmacology,Biochemistry

Reference36 articles.

1. The inhibition of ribonucleotide reductase by α-(N)-heterocyclic carboxaldehyde thiosemicarbazones;Moore,1989

2. Triapine (3-aminopyridine-2-carboxaldehyde-thiosemicarbazone): a potent inhibitor of ribonucleotide reductase activity with broad spectrum antitumor activity;Finch;Biochem Pharmacol,2000

3. Dipyridyl thiosemicarbazone chelators with potent and selective antitumor activity form iron complexes with redox activity;Richardson;J Med Chem,2006

4. The medicinal chemistry of novel iron chelators for the treatment of cancer;Kovacevic;Curr Top Med Chem,2011

5. Phase II study of 3-AP triapine in patients with recurrent or metastatic head and neck squamous cell carcinoma;Nutting;Ann Oncol,2009

Cited by 43 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Identification of FTY720 and COH29 as novel topoisomerase I catalytic inhibitors by experimental and computational studies;Bioorganic Chemistry;2024-06

2. Synthesis, crystal structure analysis, computational modelling and evaluation of anti-cervical cancer activity of novel 1,5-dicyclooctyl thiocarbohydrazone;Physical Chemistry Chemical Physics;2024

3. Inhibition of Topoisomerases by Metal Thiosemicarbazone Complexes;International Journal of Molecular Sciences;2023-07-27

4. Phenotypic Discovery of Thiocarbohydrazone with Anticancer Properties and Catalytic Inhibition of Human DNA Topoisomerase IIα;Pharmaceuticals;2023-02-23

5. Synthesis and Evaluation of Antiproliferative Activity, Topoisomerase IIα Inhibition, DNA Binding and Non-Clinical Toxicity of New Acridine–Thiosemicarbazone Derivatives;Pharmaceuticals;2022-09-02

同舟云学术

1.学者识别学者识别

2.学术分析学术分析

3.人才评估人才评估

"同舟云学术"是以全球学者为主线，采集、加工和组织学术论文而形成的新型学术文献查询和分析系统，可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容，当前同舟云学术共收录了国内外主流学术期刊6万余种，收集的期刊论文及会议论文总量共计约1.5亿篇，并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询！咨询电话：010-8811{复制后删除}0370

www.globalauthorid.com

TOP

Copyright © 2019-2024 北京同舟云网络信息技术有限公司
京公网安备11010802033243号京ICP备18003416号-3