Synthesis, crystal structure, biological evaluation, and molecular docking studies of quinoline-arylpiperazine derivative as potent α1A-adrenoceptor antagonist-Reference-Cited by-同舟云学术

Synthesis, crystal structure, biological evaluation, and molecular docking studies of quinoline-arylpiperazine derivative as potent α1A-adrenoceptor antagonist

Published:2017-02 Issue: Volume:1130 Page:895-900
ISSN:0022-2860
Container-title:Journal of Molecular Structure
language:en
Short-container-title:Journal of Molecular Structure

Author:

Xu Wei,Jiang Renwang,Yuan Mu^ORCID

Funder

Technological Innovation Project of Colleges and Universities in Guangdong Province

National Science Foundation of Guangdong Province

Postdoctoral Science Foundation of Guangzhou City

Guangzhou Industry-University Collaborative Innovation Major Projects

Guangdong Major Scientific and Technological Special Project for New Drug Development

Publisher

Elsevier BV

Subject

Inorganic Chemistry,Organic Chemistry,Spectroscopy,Analytical Chemistry

Reference30 articles.

1. Arylpiperazines for Management of Benign Prostatic Hyperplasia: Design, Synthesis, Quantitative Structure−Activity Relationships, and Pharmacokinetic Studies

2. Novel drug targets for the pharmacotherapy of benign prostatic hyperplasia (BPH)

3. Computational Study of Antagonist/α1A Adrenoceptor ComplexesObservations of Conformational Variations on the Formation of Ligand/Receptor Complexes

4. (Phenylpiperidinyl)cyclohexylsulfonamides: Development of α1a/1d-selective adrenergic receptor antagonists for the treatment of benign prostatic hyperplasia/lower urinary tract symptoms (BPH/LUTS)

5. RBx 6198: A novel α1-adrenoceptor antagonist for the treatment of benign prostatic hyperplasia

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