Identify of promising isoquinolone JNK1 inhibitors by combined application of 3D-QSAR, molecular docking and molecular dynamics simulation approaches
Author:
Funder
Chengdu University of TCM
Publisher
Elsevier BV
Subject
Inorganic Chemistry,Organic Chemistry,Spectroscopy,Analytical Chemistry
Reference44 articles.
1. JNK1: A protein kinase stimulated by UV light and Ha-Ras that binds and phosphorylates the c-Jun activation domain;Derijard;Cell,1994
2. The stress-activated protein kinase subfamily of c-Jun kinases;Kyriakis;Nature,1994
3. Small molecule JNK (c-Jun N-terminal kinase) inhibitors;Siddiqui;J. Med. Chem.,2010
4. The c-Jun N-terminal protein kinase family of mitogen-activated protein kinases (JNK MAPKs);Barr;Int. J. Biochem. Cell Biol.,2001
5. The JNK signal transduction pathway;Weston;Curr. Opin. Genet. Dev.,2002
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