Characterization of novel Checkpoint kinase 1 inhibitors by in vitro assays and in human cancer cells treated with topoisomerase inhibitors-Reference-Cited by-同舟云学术

Characterization of novel Checkpoint kinase 1 inhibitors by in vitro assays and in human cancer cells treated with topoisomerase inhibitors

Published:2011-08 Issue:7-8 Volume:89 Page:259-268
ISSN:0024-3205
Container-title:Life Sciences
language:en
Short-container-title:Life Sciences

Author:

Ferry Gilles,Studeny Aurélie,Bossard Céline,Kubara Philip M.,Zeyer Denis,Renaud Jean-Paul,Casara Patrick,de Nanteuil Guillaume,Wierzbicki Michel,Pfeiffer Bruno,Prudhomme Michelle,Leonce Stephane,Pierré Alain,Boutin Jean A.,Golsteyn Roy M.

Funder

Institut de Recherches Servier

The French Embassy in Canada Mobility Program

Alberta Cancer Foundation Pilot Funds

Alberta Innovates Technology Futures

Publisher

Elsevier BV

Subject

General Pharmacology, Toxicology and Pharmaceutics,General Biochemistry, Genetics and Molecular Biology,General Medicine

Reference60 articles.

1. A three-step synthesis from rebeccamycin of an efficient checkpoint kinase 1 inhibitor;Anizon;Eur J Med Chem,2009

2. Pathways governing the G1/S transition and their response to DNA damage;Bartek;FEBS Lett,2001

3. Breaching the DNA damage checkpoint via PF-00477736, a novel small-molecule inhibitor of checkpoint kinase 1;Blasina;Mol Cancer Ther,2008

4. Analysis of cyclin B1 and CDK activity during apoptosis induced by camptothecin treatment;Borgne;Oncogene,2006

5. Enhancement of cisplatin-induced cytotoxicity by 7-hydroxystaurosporine (UCN-01), a new G2-checkpoint inhibitor;Bunch;Clin Cancer Res,1996

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