Synthesis of cis-fused hexahydro-4aH-indeno[1,2-b]pyridines via intramolecular Ritter reaction and their conversion into tricyclic analogues of NK-1 and dopamine receptor ligands-Reference-Cited by-同舟云学术

Synthesis of cis-fused hexahydro-4aH-indeno[1,2-b]pyridines via intramolecular Ritter reaction and their conversion into tricyclic analogues of NK-1 and dopamine receptor ligands

Published:2002-05 Issue:21 Volume:58 Page:4225-4236
ISSN:0040-4020
Container-title:Tetrahedron
language:en
Short-container-title:Tetrahedron

Author:

Emelen Kristof Van,De Wit Tom,Hoornaert Georges J,Compernolle Frans

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Reference25 articles.

1. Diastereoselective Intramolecular Ritter Reaction: Generation of a Cis-Fused Hexahydro-4aH-indeno[1,2-b]pyridine Ring System with 4a,9b-Diangular Substituents

2. cis-Fused hexahydro-4aH-indeno[1,2-b]pyridines: transformation of bridgehead ester group and conversion to tricyclic analogues of NK-1 and dopamine receptor ligands

3. Discovery of a potent substance P antagonist: recognition of the key molecular determinant

4. Gem-disubstituted amino-ether based substance p antagonists

5. Phenyl-glycinol based NK1 receptor antagonists — towards the minimum pharmacophore

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