Stereoselective Transformation of 2H-1,4-Oxazin-2-ones into 2,(2),5,5-Tri- and Tetrasubstituted Analogues of cis-5-Hydroxy-2-piperidinemethanol and cis-5-Hydroxy-6-oxo-2-piperidinecarboxylic Acid-Reference-Cited by-同舟云学术

Stereoselective Transformation of 2H-1,4-Oxazin-2-ones into 2,(2),5,5-Tri- and Tetrasubstituted Analogues of cis-5-Hydroxy-2-piperidinemethanol and cis-5-Hydroxy-6-oxo-2-piperidinecarboxylic Acid

Published:2000-05 Issue:19 Volume:56 Page:3043-3051
ISSN:0040-4020
Container-title:Tetrahedron
language:en
Short-container-title:Tetrahedron

Author:

Wu Xiujuan,Dubois Kristof,Rogiers Joeri,Toppet Suzanne,Compernolle Frans,Hoornaert Georges J

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Reference12 articles.

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2. Sedum alkaloids. X. Structure and synthesis of new 3- and 5-hydroxypiperidine alkaloids

3. Alcaloïdes Pipéridiniques II. Structures de la Prosopine et de la Prosopinine, Alcaloïdes du Prosopis Africana (Guill. et Perr.) Taub. [1]

4. (a) Hirose, R.; Hamamichi, N.; Kitao, Y.; Matsuzaki, T.; Chiba, K.; Fujita, T. Bioorg. Med. Chem. Lett. 1996, 6, 2647–2650. (b) Lanciault, G.; Wolf, H. J. Pharm. Sci. 1965, 54, 84–88. (c) Portoghese, P. S.; Pazdernik, T. L. J. Med. Chem. 1968, 11, 12–15. (d) Balsamo, M.; Crotti, P.; Macchia, B.; Macchia, F. J. Med. Chem. 1973, 16, 224–227. (e) Balsamo, A.; Barili, P. L.; Gagliardi, M.; Lapucci, A.; Macchia, B.; Macchia, F. Eur. J. Med. Chem-Chim. Ther. 1982, 17, 285–289.

5. Piperidine-ether based hNK1 antagonists 1: Determination of the relative and absolute stereochemical requirements

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