Effective tuning of the arene and alkanesulfinamides for highly enantioselective synthesis of (S)-4-chlorophenylphenylmethylamine, a key intermediate for antihistamic (S)-cetirizine-Reference-Cited by-同舟云学术

Effective tuning of the arene and alkanesulfinamides for highly enantioselective synthesis of (S)-4-chlorophenylphenylmethylamine, a key intermediate for antihistamic (S)-cetirizine

Published:2003-05 Issue:22 Volume:44 Page:4195-4197
ISSN:0040-4039
Container-title:Tetrahedron Letters
language:en
Short-container-title:Tetrahedron Letters

Author:

Han Zhengxu,Krishnamurthy Dhileepkumar,Grover Paul,Fang Q.Kevin,Pflum Derek A.,Senanayake Chris H.

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Reference30 articles.

1. Synthesis and Thromboxane A2 Antagonistic Activity of ((1-Aryl(or Benzyl)-1-(benzenesulfonamido)methyl)phenyl)alkanoic Acid Derivatives.

2. An efficient synthesis of the benzhydrylpiperazine delta opioid agonist (+)-BW373U86

3. Asymmetric, Catalytic Phenyl Transfer to Imines: Highly Enantioselective Synthesis of Diarylmethylamines

4. Asymmetric synthesis of amines by nucleophilic 1,2-addition of organometallic reagents to the CN-double bond

5. Additions of Organometallic Reagents to CN Bonds: Reactivity and Selectivity

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