Chapter 32. The use of bioisosteric groups in lead optimization
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Elsevier
Reference71 articles.
1. Property-Based Design: Optimization of Drug Absorption and Pharmacokinetics
2. A practitioner's perspective of the role of quantitative structure-activity analysis in medicinal chemistry
3. The Chemistry of Pseudomonic Acid. 15. Synthesis and Antibacterial Activity of a Series of 5-Alkyl, 5-Alkenyl, and 5-Heterosubstituted Oxazoles
4. Oxadiazoles as Ester Bioisosteric Replacements in Compounds Related to Disoxaril. Antirhinovirus Activity
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