Receptor activation involving positive allosteric modulation, unlike full agonism, does not result in GABAB receptor desensitization

Author:

Gjoni Tina,Urwyler Stephan

Publisher

Elsevier BV

Subject

Cellular and Molecular Neuroscience,Pharmacology

Reference36 articles.

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4. Allosteric binding sites on cell-surface receptors: novel targets for drug discovery;Christopoulos;Nat. Rev. Drug Discov.,2002

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