Molecular Mechanism of SSR128129E, an Extracellularly Acting, Small-Molecule, Allosteric Inhibitor of FGF Receptor Signaling-Reference-Cited by-同舟云学术

Molecular Mechanism of SSR128129E, an Extracellularly Acting, Small-Molecule, Allosteric Inhibitor of FGF Receptor Signaling

Published:2013-04 Issue:4 Volume:23 Page:489-501
ISSN:1535-6108
Container-title:Cancer Cell
language:en
Short-container-title:Cancer Cell

Author:

Herbert Corentin,Schieborr Ulrich,Saxena Krishna,Juraszek Jarek,De Smet Frederik,Alcouffe Chantal,Bianciotto Marc,Saladino Giorgio,Sibrac David,Kudlinzki Denis,Sreeramulu Sridhar,Brown Alan,Rigon Patrice,Herault Jean-Pascal,Lassalle Gilbert,Blundell Tom L.,Rousseau Frederic,Gils Ann,Schymkowitz Joost,Tompa Peter,Herbert Jean-Marc,Carmeliet Peter,Gervasio Francesco Luigi,Schwalbe Harald,Bono Françoise

Publisher

Elsevier BV

Subject

Cancer Research,Cell Biology,Oncology

Reference33 articles.

1. The FGF family: biology, pathophysiology and therapy;Beenken;Nat. Rev. Drug Discov.,2009

2. Keratinocyte growth factor receptor ligands target the receptor to different intracellular pathways;Belleudi;Traffic,2007

3. Optimized molecular dynamics force fields applied to the helix-coil transition of polypeptides;Best;J. Phys. Chem. B,2009

4. Inhibition of tumor angiogenesis and growth by a small-molecule multi-FGF receptor blocker with allosteric properties;Bono;Cancer Cell,2013

5. NMR screening applied to the fragment-based generation of inhibitors of creatine kinase exploiting a new interaction proximate to the ATP binding site;Bretonnet;J. Med. Chem.,2007

Cited by 112 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Differential effects of the N‐terminal helix of FGF8b on the activity of a small‐molecule FGFR inhibitor in cell culture and for the extracellular domain of FGFR3c in solution;FEBS Letters;2024-07-12

2. A comprehensive overview of selective and novel fibroblast growth factor receptor inhibitors as a potential anticancer modality;Acta Pharmaceutica;2024-03-01

3. The Application of Artificial Intelligence and Drug Repositioning for the Identification of Fibroblast Growth Factor Receptor Inhibitors: A Review;Advanced Biomedical Research;2024-01

4. Receptor Tyrosine Kinase KIT: Mutation-Induced Conformational Shift Promotes Alternative Allosteric Pockets;Kinases and Phosphatases;2023-09-25

5. Intravitreal injection of FGF and TGF-β inhibitors disrupts cranial cartilage development;Differentiation;2023-09