Synthesis of trans-16-triazolyl-13α-methyl-17-estradiol diastereomers and the effects of structural modifications on their in vitro antiproliferative activities-Reference-Cited by-同舟云学术

Synthesis of trans-16-triazolyl-13α-methyl-17-estradiol diastereomers and the effects of structural modifications on their in vitro antiproliferative activities

Published:2015-06 Issue: Volume:150 Page:123-134
ISSN:0960-0760
Container-title:The Journal of Steroid Biochemistry and Molecular Biology
language:en
Short-container-title:The Journal of Steroid Biochemistry and Molecular Biology

Author:

Mernyák Erzsébet,Kovács Ida,Minorics Renáta,Sere Péter,Czégány Dóra,Sinka Izabella,Wölfling János,Schneider Gyula,Újfaludi Zsuzsanna,Boros Imre,Ocsovszki Imre,Varga Mónika,Zupkó István

Funder

Hungarian Scientific Research Fund

Richter Gedeon Plc

Publisher

Elsevier BV

Subject

Cell Biology,Clinical Biochemistry,Endocrinology,Molecular Biology,Molecular Medicine,Biochemistry,Endocrinology, Diabetes and Metabolism

Reference40 articles.

1. Stimulation of MCF-7 breast cancer cell proliferation by estrone sulfate and dehydroepiandrosterone sulfate: inhibition by novel non-steroidal steroid sulfatase inhibitors;Billich;J. Steroid Biochem. Mol. Biol.,2000

2. A novel steroidal selective steroid sulfatase inhibitor KW-2581 inhibits sulfated-estrogen dependent growth of breast cancer cells in vitro and in animal models;Ishida;Breast Cancer Res. Treat.,2007

3. Structure-activity relationships of C-17-substituted estratriene-3-O-sulfamates as anticancer agents;Jourdan;J. Med. Chem.,2008

4. Structure-activity relationships of 2-,4-, or 6-substituted estrogens as aromatase inhibitors;Numazawa;J. Steroid Biochem. Mol. Biol.,2005

5. C6-(N,N-butyl-methyl-heptanamide) derivatives of estrone and estradiol as inhibitors of type 1 17β-hydroxysteroid dehydrogenase: chemical synthesis and biological evaluation;Cadot;Bioorg. Med. Chem.,2007

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