In vivo potent BM635 analogue with improved drug-like properties-Reference-Cited by-同舟云学术

In vivo potent BM635 analogue with improved drug-like properties

Published:2018-02 Issue: Volume:145 Page:539-550
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Poce Giovanna^ORCID,Cocozza Martina,Alfonso Salvatore,Consalvi Sara,Venditti Giulia^ORCID,Fernandez-Menendez Raquel,Bates Robert H.,Barros Aguirre David,Ballell Lluis,De Logu Alessandro,Vistoli Giulio,Biava Mariangela

Funder

Tres Cantos Open Lab Foundation

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference18 articles.

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3. SAR analysis of new anti-TB drugs currently in pre-clinical and clinical development;Poce;Eur. J. Med. Chem.,2014

4. Bactericidal activities of the pyrrole derivative BM212 against multidrug-resistant and intramacrophagic Mycobacterium tuberculosis strains;Deidda;Antimicrob. Agents Chemother.,1998

5. 1,5-Diaryl-2-ethyl pyrrole derivatives as antimycobacterial agents: design, synthesis, and microbiological evaluation;Biava;Eur. J. Med. Chem.,2009

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