N-Phenyl indole derivatives as AT1 antagonists with anti-hypertension activities: Design, synthesis and biological evaluation-Reference-Cited by-同舟云学术

N-Phenyl indole derivatives as AT1 antagonists with anti-hypertension activities: Design, synthesis and biological evaluation

Published:2016-06 Issue: Volume:115 Page:161-178
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Zhu Weibo,Bao Xiaolu,Ren He,Da Yajing,Wu Dan,Li Fuming,Yan Yijia,Wang Li,Chen Zhilong

Funder

National Natural Science Foundation

Foundation of Shanghai Government

Foundation of Donghua University

Foundation of Ningbo Government

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference18 articles.

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3. The in vitro pharmacological profile of KR31080, a nonpeptide AT1 receptor antagonist;Hong;Fundam. Clin. Pharmacol.,1998

4. Angiotensin II type I receptor antagonist inhibits the gene expression of transforming growth factor-beta 1 and extracellular matrix in cardiac and vascular tissues of hypertensive rats;Kim;J. Pharmacol. Exp. Ther.,1995

5. Nonpeptide angiotensin II receptor antagonists. VII. Cellular and biochemical pharmacology of DuP 753, an orally active antihypertensive agent;Chiu;J. Pharmacol. Exp. Ther.,1990

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