Rational design of allosteric modulators of the aromatase enzyme: An unprecedented therapeutic strategy to fight breast cancer-Reference-Cited by-同舟云学术

Rational design of allosteric modulators of the aromatase enzyme: An unprecedented therapeutic strategy to fight breast cancer

Published:2019-04 Issue: Volume:168 Page:253-262
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Spinello Angelo^ORCID,Martini Silvia,Berti Federico^ORCID,Pennati Marzia,Pavlin Matic,Sgrignani Jacopo^ORCID,Grazioso Giovanni^ORCID,Colombo Giorgio,Zaffaroni Nadia,Magistrato Alessandra^ORCID

Funder

Italian Association For Cancer Research

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference90 articles.

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3. Influence of the membrane lipophilic environment on the structure and on the substrate access/egress routes of the human aromatase enzyme. A computational study;Sgrignani;J. Chem. Inf. Model.,2012

4. A dehydrogenase dual hydrogen abstraction mechanism promotes estrogen biosynthesis: can we expand the functional annotation of the aromatase enzyme?;Spinello;Chem. Eur J.,2018

5. Estrogen receptor alpha-36 (ER-alpha36): a new player in human breast cancer;Wang;Mol. Cell. Endocrinol.,2015

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