Design, synthesis and bioevaluation of N-trisubstituted pyrimidine derivatives as potent aurora A kinase inhibitors
Author:
Funder
Guangdong Innovative Research Team Program
The National High-tech R&D Program of China
Publisher
Elsevier BV
Subject
Organic Chemistry,Drug Discovery,Pharmacology,General Medicine
Reference25 articles.
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3. Aurora kinase inhibitors in preclinical and clinical testing;Cheung;Expert Opinion on Investigational Drugs,2009
4. ENMD-2076 is an orally active kinase inhibitor with antiangiogenic and antiproliferative mechanisms of action;Fletcher;Molecular Cancer Therapeutics,2011
5. Discovery of N-phenyl-4-(thiazol-5-yl)pyrimidin-2-amine aurora kinase inhibitors;Wang;Journal of Medicinal Chemistry,2010
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