New N -phenylpyrrolamide DNA gyrase B inhibitors: Optimization of efficacy and antibacterial activity

Author:

Durcik Martina,Lovison Denise,Skok Žiga,Durante Cruz Cristina,Tammela PäiviORCID,Tomašič TihomirORCID,Benedetto Tiz Davide,Draskovits Gábor,Nyerges Ákos,Pál Csaba,Ilaš JanezORCID,Peterlin Mašič Lucija,Kikelj Danijel,Zidar NaceORCID

Funder

Slovenian Research Agency

Academy of Finland

European Research Council

Hungarian Academy of Sciences

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference43 articles.

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2. Thiophene antibacterials that allosterically stabilize DNA-cleavage complexes with DNA gyrase;Chan;Proc. Natl. Acad. Sci. U. S. A,2017

3. Bad bugs, no drugs: no ESKAPE! an update from the Infectious Diseases Society of America;Boucher;Clin. Infect. Dis.,2009

4. Global priority list of antibiotic-resistant to guide research, discovery, and development of new antibiotics;World Health Organisation,2017

5. Exploiting bacterial DNA gyrase as a drug target: current state and perspectives;Collin;Appl. Microbiol. Biotechnol.,2011

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