New <i>N</i>-phenylpyrrolamide inhibitors of DNA gyrase with improved antibacterial activity-Reference-Cited by-同舟云学术

New N-phenylpyrrolamide inhibitors of DNA gyrase with improved antibacterial activity

Published:2024 Issue:39 Volume:14 Page:28423-28454
ISSN:2046-2069
Container-title:RSC Advances
language:en
Short-container-title:RSC Adv.

Author:

Cotman Andrej Emanuel¹^ORCID,Fulgheri Federica¹,Piga Martina¹^ORCID,Peršolja Peter¹^ORCID,Tiz Davide Benedetto¹^ORCID,Skok Žiga¹^ORCID,Durcik Martina¹,Sterle Maša¹,Dernovšek Jaka¹^ORCID,Cruz Cristina D.²,Tammela Päivi²^ORCID,Szili Petra Éva³,Daruka Lejla³,Pál Csaba³,Zega Anamarija¹,Mašič Lucija Peterlin¹,Ilaš Janez¹^ORCID,Tomašič Tihomir¹^ORCID,Kikelj Danijel¹,Zidar Nace¹^ORCID

Affiliation:

1. University of Ljubljana, Faculty of Pharmacy, Aškerčeva cesta 7, 1000 Ljubljana, Slovenia

2. Drug Research Program, Division of Pharmaceutical Biosciences, Faculty of Pharmacy, University of Helsinki, P.O. Box 56, Viikinkaari 5E, Helsinki 00014, Finland

3. Synthetic and Systems Biology Unit, Institute of Biochemistry, Biological Research Centre of the Hungarian Academy of Sciences, Szeged, H-6726, Hungary

Abstract

New N-phenylpyrrolamide inhibitors of DNA gyrase were developed with excellent on-target activity and improved antibacterial activity.

Funder

Javna Agencija za Raziskovalno Dejavnost RS

Research Council of Finland

Nemzeti Kutatási Fejlesztési és Innovációs Hivatal

Publisher

Royal Society of Chemistry (RSC)

Link

http://pubs.rsc.org/en/content/articlepdf/2024/RA/D4RA04802D

Reference38 articles.

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