Synthesis of novel galeterone derivatives and evaluation of their in vitro activity against prostate cancer cell lines-Reference-Cited by-同舟云学术

Synthesis of novel galeterone derivatives and evaluation of their in vitro activity against prostate cancer cell lines

Published:2019-10 Issue: Volume:179 Page:483-492
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Jorda Radek^ORCID,Řezníčková Eva,Kiełczewska Urszula,Maj Jadwiga,Morzycki Jacek W.,Siergiejczyk Leszek,Bazgier Václav^ORCID,Berka Karel^ORCID,Rárová Lucie^ORCID,Wojtkielewicz Agnieszka^ORCID

Funder

Palacký University in Olomouc

Czech Science Foundation

European Regional Development

Polish National Science Centre

ELIXIR CZ research infrastructure project

Operational Programme Research, Development and Education – European Regional Development

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference17 articles.

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2. Androgen receptor targeted treatments of prostate cancer: 35 Years of progress with antiandrogens;Crawford;J. Urol.,2018

3. AR-V7 and resistance to enzalutamide and abiraterone in prostate cancer;Antonarakis;N. Engl. J. Med.,2014

4. Galeterone for the treatment of advanced prostate cancer: the evidence to date;Bastos;Drug Des. Dev. Ther.,2016

5. Novel galeterone analogs act independently of AR and AR-V7 for the activation of the unfolded protein response and induction of apoptosis in the CWR22Rv1 prostate cancer cell model;McCarty;Oncotarget,2017

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