Discovery of 4-aminoquinolines as highly selective TGFβR1 inhibitors with an attenuated MAP4K4 profile for potential applications in immuno-oncology-Reference-Cited by-同舟云学术

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Discovery of 4-aminoquinolines as highly selective TGFβR1 inhibitors with an attenuated MAP4K4 profile for potential applications in immuno-oncology

Published:2021-12 Issue: Volume:225 Page:113763
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Kharbanda Anupreet,Tran Phuc,Zhang Lingtian,Leung Yuet-Kin,Li Hong-yu,Frett Brendan

Funder

National Institutes of Health

National Institute of General Medical Sciences

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference50 articles.

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2. The immune system and cancer evasion strategies: therapeutic concepts;Muenst;J. Intern. Med.,2016

3. Immune evasion in cancer: mechanistic basis and therapeutic strategies;Vinay;Semin. Canc. Biol.,2015

4. The immunobiology of cancer immunosurveillance and immunoediting;Dunn;Immunity,2004

5. Immune checkpoint inhibitors: recent progress and potential biomarkers;Darvin;Exp. Mol. Med.,2018

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1. Advances in the discovery of activin receptor-like kinase 5 (ALK5) inhibitors;Bioorganic Chemistry;2024-06

2. Design, Synthesis, and In Vitro Antiproliferative Activity of 4,5,6-Trisubstituted 2-Aminopyrimidines as Potential TGF-β Inhibitors;Russian Journal of Organic Chemistry;2024-04

3. Metal-free [2 + 2] and [4 + 2] cycloadditions ofN-aryl-substituted ynamides to construct functionalized aminocyclobutenes and 4-aminoquinolines;Organic Chemistry Frontiers;2023

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