Design, synthesis and biological evaluation of sulfamoylphenyl-quinazoline derivatives as potential EGFR/CAIX dual inhibitors
Author:
Publisher
Elsevier BV
Subject
Organic Chemistry,Drug Discovery,Pharmacology,General Medicine
Reference55 articles.
1. Discovery of potent and selective epidermal growth factor receptor (EGFR) bifunctional small-molecule degraders;Cheng;J. Med. Chem.,2020
2. Kahksha, M.T. Alam, M. Imran, Novel quinazoline-based EGFR kinase inhibitors: a review focussing on SAR and molecular docking studies (2015-2019),;Bhatia;Eur. J. Med. Chem.,2020
3. Contemporary challenges in the design of topoisomerase II inhibitors for cancer chemotherapy;Bailly;Chem. Rev.,2012
4. Polypharmacology: challenges and opportunities in drug discovery;Anighoro;J. Med. Chem.,2014
5. De novo design of multitarget ligands with an iterative fragment-growing strategy;Shang;J. Chem. Inf. Model.,2014
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