Chemoenzymatic synthesis of 2,6-disubstituted tetrahydropyrans with high σ1 receptor affinity, antitumor and analgesic activity-Reference-Cited by-同舟云学术

Chemoenzymatic synthesis of 2,6-disubstituted tetrahydropyrans with high σ1 receptor affinity, antitumor and analgesic activity

Published:2021-07 Issue: Volume:219 Page:113443
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Kopp Nicole,Civenni Gianluca^ORCID,Marson Domenico,Laurini Erik,Pricl Sabrina^ORCID,Catapano Carlo V.^ORCID,Humpf Hans-Ulrich^ORCID,Almansa Carmen,Nieto Francisco Rafael,Schepmann Dirk,Wünsch Bernhard^ORCID

Funder

Deutsche Forschungsgemeinschaft

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference75 articles.

1. The effects of morphine- and nalorphine- like drugs in the nondependent and morphine-dependent chronic spinal dog;Martin;J. Pharmacol. Exp. Therapeut.,1976

2. Naltrexone fails to antagonize the σ-effects of PCP and SKF 10,047 in the dog;Vaupel;Eur. J. Pharmacol.,1983

3. A sigma-like binding site in rat pheochromocytoma (PC12) cells: decreased affinity for (+)-benzomorphans and lower molecular weight suggest a different sigma receptor form from that of Guinea pig brain;Hellewell;Brain Res.,1990

4. Rat liver and kidney contain high densities of sigma 1 and sigma 2 receptors: characterization by ligand binding and photoaffinity labeling;Hellewell;Eur. J. Pharmacol.,1994

5. Sigma receptors Are associated with cortical Limbic areas in the primate brain;Mash;Synapse,1992

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