Design, synthesis and biological evaluation of novel thiazolidinedione derivatives as irreversible allosteric IKK-β modulators-Reference-Cited by-同舟云学术

Design, synthesis and biological evaluation of novel thiazolidinedione derivatives as irreversible allosteric IKK-β modulators

Published:2018-09 Issue: Volume:157 Page:691-704
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Elkamhawy Ahmed^ORCID,Kim Nam youn,Hassan Ahmed H.E.^ORCID,Park Jung-eun,Yang Jeong-Eun,Oh Kwang-Seok,Lee Byung Ho,Lee Mi Young,Shin Kye Jung,Lee Kyung-Tae,Hur Wooyoung,Roh Eun Joo^ORCID

Funder

KIST

National Research Council of Science & Technology

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference34 articles.

1. Chapter 3 the learning and evolution of medicinal chemistry against kinase targets;Swarbrick,2012

2. The regulation of protein function by multisite phosphorylation – a 25 year update;Cohen;Trends Biochem. Sci.,2000

3. Kinase selectivity potential for inhibitors targeting the ATP binding site: a network analysis;Huang;Bioinformatics,2010

4. Strategies for the selective regulation of kinases with allosteric modulators: exploiting exclusive structural features;Fang;ACS Chem. Biol.,2013

5. CHAPTER 3 targeting catalytic and non-catalytic functions of protein kinases;Muller,2017

Cited by 23 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Design, synthesis, and evaluation of new anti-inflammatory natural products amide derivatives endowed with anti-blood cancer activity towards development of potential multifunctional agents against hematological cancers;European Journal of Medicinal Chemistry;2023-10

2. Design, synthesis, and study of novel phenethyl-based antitumor phospholipids downregulating p38 mitogen-activated protein kinase;Journal of Enzyme Inhibition and Medicinal Chemistry;2023-05-29

3. Chemistry and Applications of Functionalized 2,4‐Thiazolidinediones;European Journal of Organic Chemistry;2023-05-03

4. The anti-inflammatory activity of 2-iminothiazolidines: evidence for macrophage repolarization;Inflammopharmacology;2022-10-22

5. From EGFR kinase inhibitors to anti-inflammatory drugs: Optimization and biological evaluation of (4-(phenylamino)quinazolinyl)-phenylthiourea derivatives as novel NF-κB inhibitors;Bioorganic Chemistry;2022-10