[1,2,4]Triazolo[1,5-c]pyrimidines as adenosine receptor antagonists: Modifications at the 8 position to reach selectivity towards A3 adenosine receptor subtype-Reference-Cited by-同舟云学术

[1,2,4]Triazolo[1,5-c]pyrimidines as adenosine receptor antagonists: Modifications at the 8 position to reach selectivity towards A3 adenosine receptor subtype

Published:2018-09 Issue: Volume:157 Page:837-851
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Federico Stephanie^ORCID,Margiotta Enrico,Salmaso Veronica,Pastorin Giorgia,Kachler Sonja,Klotz Karl-Norbert,Moro Stefano^ORCID,Spalluto Giampiero

Funder

NVIDIA Corporation

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference39 articles.

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3. International union of basic and clinical pharmacology. LXXXI. Nomenclature and classification of adenosine receptors — an update;Fredholm;Pharmacol. Rev.,2011

4. Adenosine receptors as therapeutic targets;Jacobson;Nat. Rev. Drug Discov.,2006

5. Cardio-renal effects of the A1 adenosine receptor antagonist SLV320 in patients with heart failure;Mitrovic;Circ. Hear. Fail,2009

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