A chemical perspective on the modulation of TEAD transcriptional activities: Recent progress, challenges, and opportunities
Author:
Publisher
Elsevier BV
Subject
Organic Chemistry,Drug Discovery,Pharmacology,General Medicine
Reference198 articles.
1. MST1/MST2 protein kinases: regulation and physiologic roles;Galan;Biochemistry,2016
2. The Ste20-like kinase Mst2 activates the human large tumor suppressor kinase Lats1;Chan;Oncogene,2005
3. A coordinated phosphorylation by Lats and CK1 regulates YAP stability through SCF(beta-TRCP);Zhao;Genes Dev.,2010
4. Elucidation of a universal size-control mechanism in drosophila and mammals;Dong;Cell,2007
5. Inactivation of YAP oncoprotein by the Hippo pathway is involved in cell contact inhibition and tissue growth control;Zhao;Genes Dev.,2007
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2. Design, Synthesis, and Bioevaluation of Transcriptional Enhanced Assocciated Domain (TEAD) PROTAC Degraders;ACS Medicinal Chemistry Letters;2024-04-22
3. Allosteric Modulation of the YAP/TAZ-TEAD Interaction by Palmitoylation and Small-Molecule Inhibitors;The Journal of Physical Chemistry B;2024-04-12
4. TRIM21 is critical in regulating hepatocellular carcinoma growth and response to therapy by altering the MST1/YAP pathway;Cancer Science;2024-03-12
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