New thiazole-based derivatives as EGFR/HER2 and DHFR inhibitors: Synthesis, molecular modeling simulations and anticancer activity
Author:
Publisher
Elsevier BV
Subject
Organic Chemistry,Drug Discovery,Pharmacology,General Medicine
Reference53 articles.
1. Inhibitor of ovarian cancer cells growth by virtual screening: a new thiazole derivative targeting human thymidylate synthase;Carosati;J. Med. Chem.,2012
2. Molecular modelling and biological evaluation of tetrasubstituted thiazoles towards cholinesterase enzymes and cytotoxicity studies;Mumtaz;Bioorg. Chem.,2018
3. Antibacterial, antibiofilm and molecular modeling study of some antitumor thiazole based chalcones as a new class of DHFR inhibitors;Alrohily;Microb. Pathog.,2019
4. Discovery of a novel DNA polymerase inhibitor and characterization of its antiproliferative properties;Mishra;Cancer Biol. Ther.,2019
5. Tyrosine kinase inhibitors for solid tumors in the past 20 years (2001–2020);Huang;J. Hematol. Oncol.,2020
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