Discovery of potent and highly selective covalent inhibitors of Bruton’s tyrosine kinase bearing triazine scaffold-Reference-Cited by-同舟云学术

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Discovery of potent and highly selective covalent inhibitors of Bruton’s tyrosine kinase bearing triazine scaffold

Published:2020-08 Issue: Volume:199 Page:112339
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Teng Yu,Lu Xiang,Xiao Maoxu,Li Zhenbang,Zou Yumei,Ren Shengnan,Cheng Yu,Luo Guoshun,Xiang Hua

Funder

Program of Jiangsu Key Laboratory of Drug Design and Optimization, China Pharmaceutical University

Natural Science Foundation of China

NSFC

CPU

College students’ innovation and entrepreneurship training program

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference30 articles.

1. Targeting Bruton’s tyrosine kinase with ibrutinib in B-cell malignancies;Wang;Clin. Pharmacol. Therapeut.,2015

2. The B cell receptor signaling pathway in mantle cell lymphoma;Merolle;Oncotarget,2018

3. Design and synthesis of sulfonamide-substituted diphenylpyrimidines (SFA-DPPYs) as potent Bruton’s tyrosine kinase (BTK) inhibitors with improved activity toward B-cell lymphoblastic leukemia;Liu;Eur. J. Med. Chem.,2017

4. Discovery and structure-activity relationship of novel diphenylthiazole derivatives as BTK inhibitor with potent activity against B cell lymphoma cell lines;Guo;Eur. J. Med. Chem.,2019

5. Discovery of a series of 2,5-diaminopyrimidine covalent irreversible inhibitors of Bruton’s tyrosine kinase with in vivo antitumor activity;Li;J. Med. Chem.,2014

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