Structural modifications in the distal, regulatory region of histamine H3 receptor antagonists leading to the identification of a potent anti-obesity agent-Reference-Cited by-同舟云学术

Structural modifications in the distal, regulatory region of histamine H3 receptor antagonists leading to the identification of a potent anti-obesity agent

Published:2021-03 Issue: Volume:213 Page:113041
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Szczepańska Katarzyna,Pockes Steffen^ORCID,Podlewska Sabina,Höring Carina,Mika Kamil,Latacz Gniewomir,Bednarski Marek,Siwek Agata,Karcz Tadeusz,Nagl Martin,Bresinsky Merlin,Mönnich Denise,Seibel Ulla^ORCID,Kuder Kamil J.,Kotańska Magdalena,Stark Holger,Elz Sigurd^ORCID,Kieć-Kononowicz Katarzyna

Funder

Deutsche Forschungsgemeinschaft

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference54 articles.

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5. Progress in the development of histamine H3 receptor antagonists/inverse agonists: a patent review (2013-2017);Łażewska;Expert Opin. Ther. Pat.,2018

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1. The Effect of KSK-94, a Dual Histamine H3 and Sigma-2 Receptor Ligand, on Adipose Tissue in a Rat Model of Developing Obesity;Pharmaceuticals;2024-07-01

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4. Evaluation of Some Safety Parameters of Dual Histamine H3 and Sigma-2 Receptor Ligands with Anti-Obesity Potential;International Journal of Molecular Sciences;2023-04-19

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