Dual Piperidine-Based Histamine H3 and Sigma-1 Receptor Ligands in the Treatment of Nociceptive and Neuropathic Pain

Author:

Szczepańska Katarzyna12ORCID,Karcz Tadeusz1,Dichiara Maria3ORCID,Mogilski Szczepan4,Kalinowska-Tłuścik Justyna5,Pilarski Bogusław6,Leniak Arkadiusz7,Pietruś Wojciech27ORCID,Podlewska Sabina2ORCID,Popiołek-Barczyk Katarzyna8,Humphrys Laura J.9ORCID,Ruiz-Cantero M. Carmen10ORCID,Reiner-Link David11,Leitzbach Luisa11,Łażewska Dorota1ORCID,Pockes Steffen9ORCID,Górka Michał7,Zmysłowski Adam7,Calmels Thierry12,Cobos Enrique J.10,Marrazzo Agostino3ORCID,Stark Holger11ORCID,Bojarski Andrzej J.2ORCID,Amata Emanuele3ORCID,Kieć-Kononowicz Katarzyna1

Affiliation:

1. Department of Technology and Biotechnology of Drugs, Faculty of Pharmacy, Jagiellonian University Medical College, Medyczna 9, 30-688 Kraków, Poland

2. Department of Medicinal Chemistry, Maj Institute of Pharmacology, Polish Academy of Sciences, Smętna 12, 31-343 Kraków, Poland

3. Department of Drug and Health Sciences, University of Catania, V.le A. Doria, 95125 Catania, Italy

4. Department of Pharmacodynamics, Faculty of Pharmacy, Jagiellonian University Medical College, Medyczna 9, 30-688 Kraków, Poland

5. Department of Crystal Chemistry and Crystal Physics, Faculty of Chemistry, Jagiellonian University, Gronostajowa 2, 30-387 Kraków, Poland

6. Cerko Sp. z o.o. Sp.k, Al. Zwycięstwa 96/98, 81-451 Gdynia, Poland

7. Celon Pharma S.A., R&D Centre, Marymoncka 15, 05-152 Kazuń Nowy, Poland

8. Department of Neurochemistry, Maj Institute of Pharmacology, Polish Academy of Sciences, Smętna 12, 31-343 Kraków, Poland

9. Institute of Pharmacy, Faculty of Chemistry and Pharmacy, University of Regensburg, Universitätsstraße 31, D-93053 Regensburg, Germany

10. Department of Pharmacology and Neurosciences Institute (Biomedical Research Center), University of Granada, and Biosanitary Research Institute ibs. Granada, Avenida de la Investigación 11, 18016 Granada, Spain

11. Institute of Pharmaceutical and Medicinal Chemistry, Heinrich Heine University Düsseldorf, Universitaetsstr. 1, 40225 Düsseldorf, Germany

12. Bioprojet-Biotech, 4rue du Chesnay Beauregard, 35762 Saint-Gregoire Cedex, France

Funder

Ministerstwo Edukacji i Nauki

Universit? di Catania

Uniwersytet Jagiellonski Collegium Medicum

Narodowe Centrum Nauki

Deutsche Forschungsgemeinschaft

European Cooperation in Science and Technology

Fonds der Chemischen Industrie

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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