Flexible diaminodihydrotriazine inhibitors of Plasmodium falciparum dihydrofolate reductase: Binding strengths, modes of binding and their antimalarial activities-Reference-Cited by-同舟云学术

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Flexible diaminodihydrotriazine inhibitors of Plasmodium falciparum dihydrofolate reductase: Binding strengths, modes of binding and their antimalarial activities

Published:2020-06 Issue: Volume:195 Page:112263
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Kamchonwongpaisan Sumalee,Charoensetakul Netnapa,Srisuwannaket Choladda,Taweechai Supannee,Rattanajak Roonglawan,Vanichtanankul Jarunee,Vitsupakorn Danoo,Arwon Uthai,Thongpanchang Chawanee,Tarnchompoo Bongkoch,Vilaivan Tirayut,Yuthavong Yongyuth

Funder

UNICEF/World Bank/World Health Organization/Special Program in Tropical Diseases

Medicines for Malaria Venture

BIOTEC

NSTDA’s Cluster and Program Management

NSTDA’s Researcher Chair Grant

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference55 articles.

1. Amino acid changes linked to pyrimethamine resistance in the dihydrofolate reductase–thymidylate synthase gene of Plasmodium falciparum;Cowman;Proc. Natl. Acad. Sci. U.S.A.,1988

2. Resistance to antifolates in Plasmodium falciparum monitored by sequence analysis of dihydropteroate synthetase and dihydrofolate reductase alleles in a large number of field samples of diverse origins;Wang;Mol. Biochem. Parasitol.,1997

3. P. falciparum dihydrofolate reductase and dihydropteroate synthase mutations: epidemiology and role in clinical resistance to antifolates;Plowe;Drug Resist. Updates,1998

4. Evidence that a point mutation in dihydrofolate reductase-thymidylate synthase confers resistance to pyrimethamine in falciparum malaria;Peterson;Proc. Natl. Acad. Sci. U.S.A.,1988

5. Molecular basis of differential resistance to cycloguanil and pyrimethamine in Plasmodium falciparum malaria;Peterson;Proc. Natl. Acad. Sci. U.S.A.,1990

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