Development of bivalent triarylalkene- and cyclofenil-derived dual estrogen receptor antagonists and downregulators-Reference-Cited by-同舟云学术

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Development of bivalent triarylalkene- and cyclofenil-derived dual estrogen receptor antagonists and downregulators

Published:2020-04 Issue: Volume:192 Page:112191
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Knox Alexandra,Kalchschmid Christina,Schuster Daniela,Gaggia Francesca,Manzl Claudia,Baecker Daniel,Gust Ronald

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference58 articles.

1. Antiestrogens and selective estrogen receptor modulators as multifunctional medicines. 1. Receptor interactions;Jordan;J. Med. Chem.,2003

2. Antiestrogens and selective estrogen receptor modulators as multifunctional medicines. 2. Clinical considerations and new agents;Jordan;J. Med. Chem.,2003

3. Design, synthesis, and in vitro biological evaluation of small molecule inhibitors of estrogen receptor alpha coactivator binding;Rodriguez;J. Med. Chem.,2004

4. Discovering small-molecule estrogen receptor alpha/coactivator binding inhibitors: high-throughput screening, ligand development, and models for enhanced potency;Sun;ChemMedChem,2011

5. Recent advances in peptidomimetics antagonists targeting estrogen receptor alpha-coactivator interaction in cancer therapy;Qin;Bioorg. Med. Chem. Lett.,2018

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1. Development of Cytotoxic GW7604-Zeise’s Salt Conjugates as Multitarget Compounds with Selectivity for Estrogen Receptor- Positive Tumor Cells;Journal of Medicinal Chemistry;2024-03-13

2. Development of heterodimeric estrogen receptor alpha antagonists to target simultaneously the ligand and coactivator binding site;Archiv der Pharmazie;2023-05-12

3. DNA-modularized construction of bivalent ligands precisely regulates receptor binding and activation;Chem;2023-04

4. Rational design, synthesis, antiproliferative activity against MCF-7, MDA-MB-231 cells, estrogen receptors binding affinity, and computational study of indenopyrimidine-2,5-dione analogs for the treatment of breast cancer;Bioorganic & Medicinal Chemistry Letters;2022-05

5. Structure-based design and synthesis of conformationally constrained derivatives of methyl-piperidinopyrazole (MPP) with estrogen receptor (ER) antagonist activity;Bioorganic Chemistry;2022-02

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