Design, Synthesis, and in Vitro Biological Evaluation of Small Molecule Inhibitors of Estrogen Receptor α Coactivator Binding
Author:
Affiliation:
1. Department of Chemistry, University of Illinois, 600 South Mathews Avenue, Urbana, Illinois 61801
Publisher
American Chemical Society (ACS)
Subject
Drug Discovery,Molecular Medicine
Link
https://pubs.acs.org/doi/pdf/10.1021/jm030404c
Reference48 articles.
1. Minireview: Nuclear Receptor Coactivators—An Update
2. Combinatorial Control of Gene Expression by Nuclear Receptors and Coregulators
3. The Structural Basis of Estrogen Receptor/Coactivator Recognition and the Antagonism of This Interaction by Tamoxifen
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