Novel 2,3-disubstituted quinazoline-4(3 H )-one molecules derived from amino acid linked sulphonamide as a potent malarial antifolates for DHFR inhibition-Reference-Cited by-同舟云学术

Novel 2,3-disubstituted quinazoline-4(3 H )-one molecules derived from amino acid linked sulphonamide as a potent malarial antifolates for DHFR inhibition

Published:2017-03 Issue: Volume:129 Page:251-265
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Patel Tarosh S.,Vanparia Satish F.,Patel Urmila H.,Dixit Ritu B.,Chudasama Chaitanya J.,Patel Bhavesh D.,Dixit Bharat C.

Funder

University Grants Commission

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference55 articles.

1. WHO, reportWorld Malaria Report 2015, World Health Organization 2015.

2. Towards an understanding of drug resistance in malaria: three-dimensional structure of Plasmodium falciparum dihydrofolate reductase by homology building;Lemcke;Bioorg. Med. Chem.,1999

3. Drug resistance in malaria parasites of animals and man;Peters;Adv. Parasitol.,1998

4. The mode of action and the mechanism of resistance to antimalarial drugs;Foote;Acta Trop.,1994

5. MALARIA: new developments in treatment and prevention;Newton;Annu. Rev. Med.,1999

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