Chromenone derivatives as a versatile scaffold with dual mode of inhibition of HIV-1 reverse transcriptase-associated Ribonuclease H function and integrase activity-Reference-Cited by-同舟云学术

Chromenone derivatives as a versatile scaffold with dual mode of inhibition of HIV-1 reverse transcriptase-associated Ribonuclease H function and integrase activity

Published:2019-11 Issue: Volume:182 Page:111617
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Esposito Francesca,Ambrosio Francesca Alessandra,Maleddu Rita,Costa Giosuè,Rocca Roberta^ORCID,Maccioni Elias^ORCID,Catalano Raffaella,Romeo Isabella,Eleftheriou Phaedra,Karia Denish C.,Tsirides Petros,Godvani Nilesh,Pandya Hetal,Corona Angela,Alcaro Stefano^ORCID,Artese Anna^ORCID,Geronikaki Athina^ORCID,Tramontano Enzo

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

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5. Biochemical characterization of a multi-drug resistant HIV-1 subtype AG reverse transcriptase: antagonism of AZT discrimination and excision pathways and sensitivity to RNase H inhibitors;Schneider;Nucleic Acids Res.,2016

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