From random to rational: A discovery approach to selective subnanomolar inhibitors of human carbonic anhydrase IV based on the Castagnoli-Cushman multicomponent reaction-Reference-Cited by-同舟云学术

From random to rational: A discovery approach to selective subnanomolar inhibitors of human carbonic anhydrase IV based on the Castagnoli-Cushman multicomponent reaction

Published:2019-11 Issue: Volume:182 Page:111642
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Kalinin Stanislav,Nocentini Alessio^ORCID,Kovalenko Alexander,Sharoyko Vladimir,Bonardi Alessandro,Angeli Andrea^ORCID,Gratteri Paola,Tennikova Tatiana B.,Supuran Claudiu T.^ORCID,Krasavin Mikhail^ORCID

Funder

Russian Federation Government

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference73 articles.

1. Structure and function of carbonic anhydrases;Supuran;Biochem. J.,2016

2. Multiple binding modes of inhibitors to carbonic anhydrases: how to design specific drugs targeting 15 different isoforms?;Alterio;Chem. Rev.,2012

3. Carbonic anhydrase inhibitors and activators for novel therapeutic applications;Supuran;Future Med. Chem.,2011

4. Diuretics: from classical carbonic anhydrase inhibitors to novel applications of the sulfonamides;Supuran;Curr. Pharmaceut. Des.,2008

5. The development of topically acting carbonic anhydrase inhibitors as antiglaucoma agents;Supuran;Curr. Pharmaceut. Des.,2008

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