[1,2,3]Triazolo[4,5-d]pyrimidine derivatives incorporating (thio)urea moiety as a novel scaffold for LSD1 inhibitors-Reference-Cited by-同舟云学术

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[1,2,3]Triazolo[4,5-d]pyrimidine derivatives incorporating (thio)urea moiety as a novel scaffold for LSD1 inhibitors

Published:2020-02 Issue: Volume:187 Page:111989
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Li Zhong-Hua^ORCID,Ma Jin-Lian,Liu Gai-Zhi,Zhang Xin-Hui,Qin Ting-Ting,Ren Wei-Hong,Zhao Tao-Qian,Chen Xiao-Hui,Zhang Zhen-Qiang

Funder

PhD Research Startup Foundation of Henan University of Chinese Medicine

Colleges and Universities Key Scientific Research Project Plan (Basic Research Special) of Henan Province

Science and Technology Project for Tackling Key Problems of Henan province

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference42 articles.

1. Histone onco-modifications;Fullgrabe;Oncogene,2011

2. Histone demethylation mediated by the nuclear amine oxidase homolog LSD1;Shi;Cell,2004

3. LSD1 demethylates repressive histone marks to promote androgen-receptor-dependent transcription;Metzger;Nature,2005

4. Histone methylation-dependent mechanisms impose ligand dependency for gene activation by nuclear receptors;Garcia-Bassets;Cell,2007

5. Chromatin remodeling and cancer, part I: covalent histone modifications;Wang;Trends Mol. Med.,2007

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2. Lysine-Specific Demethylase 1 Inhibitors: A Comprehensive Review Utilizing Computer-Aided Drug Design Technologies;Molecules;2024-01-22

3. A Quinquennial Review of Potent LSD1 Inhibitors Explored for the Treatment of Different Cancers, with Special Focus on SAR Studies;Current Medicinal Chemistry;2024-01

4. Design, synthesis and in vitro/in vivo anticancer activity of tranylcypromine-based triazolopyrimidine analogs as novel LSD1 inhibitors;European Journal of Medicinal Chemistry;2023-05

5. An Appraisal on Synthetic and Medicinal Aspects of Fused Pyrimidines as Anti Neoplastic Agents;Anti-Cancer Agents in Medicinal Chemistry;2023-03

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