Design, synthesis and in vitro/in vivo anticancer activity of tranylcypromine-based triazolopyrimidine analogs as novel LSD1 inhibitors-Reference-Cited by-同舟云学术

Design, synthesis and in vitro/in vivo anticancer activity of tranylcypromine-based triazolopyrimidine analogs as novel LSD1 inhibitors

Published:2023-05 Issue: Volume:253 Page:115321
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Li Zhonghua^ORCID,Yuan Yong,Wang Pan,Zhang Zijuan,Ma Huifen,Sun Yiran,Zhang Xiaowei,Li Xiaofang,Qiao Yonghui,Zhang Feiyu,Su Yunfang,Song Junying,Xie Zhishen,Li Lixin,Ma Liying,Ma Jinlian,Zhang Zhenqiang

Funder

Henan University of Chinese Medicine

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference27 articles.

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3. High-resolution profiling of histone methylations in the human genome;Barski;Cell,2007

4. Antagonistic actions of Rcor proteins regulate LSD1 activity and cellular differentiation;Upadhyay;P. Natl. Acad. Sci. USA.,2014

5. The lysine demethylase LSD1 (KDM1) is required for maintenance of global DNA methylation;Wang;Nat. Genet.,2009

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