Identification of potent triazolylpyridine nicotinamide phosphoribosyltransferase (NAMPT) inhibitors bearing a 1,2,3-triazole tail group-Reference-Cited by-同舟云学术

Identification of potent triazolylpyridine nicotinamide phosphoribosyltransferase (NAMPT) inhibitors bearing a 1,2,3-triazole tail group

Published:2019-11 Issue: Volume:181 Page:111576
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Travelli Cristina^ORCID,Aprile Silvio^ORCID,Mattoteia Daiana,Colombo Giorgia,Clemente Nausicaa,Scanziani Eugenio,Terrazzino Salvatore,Alisi Maria Alessandra,Polenzani Lorenzo,Grosa Giorgio,Genazzani Armando A.,Tron Gian Cesare,Galli Ubaldina^ORCID

Funder

FIRC fellowship

AIRC

Fondazione Umberto Veronesi

Angelini S.p.A

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference51 articles.

1. The NAD metabolome--a key determinant of cancer cell biology;Chiarugi;Nat. Rev. Cancer,2012

2. For an exhaustive review covering NAMPT inhibitors discovered until 2012 see

3. Medicinal chemistry of nicotinamide phosphoribosyltransferase (NAMPT) inhibitors;Galli;J. Med. Chem.,2013

4. Structure based design of nicotinamide phosphoribosyltransferase (NAMPT) inhibitors from a phenotypic screen;Palacios;Bioorg. Med. Chem. Lett,2018

5. Discovery of a highly selective NAMPT inhibitor that demonstrates robust efficacy and improved retinal toxicity with nicotinic acid coadministration;Zhao;Mol. Cancer Ther.,2017

Cited by 17 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. New Analogues of the Nicotinamide Phosphoribosyltransferase Inhibitor FK866 as Potential Anti-Pancreatic Cancer Agents;Medicinal Chemistry;2024-08

2. Design of FK866-Based Degraders for Blocking the Nonenzymatic Functions of Nicotinamide Phosphoribosyltransferase;Journal of Medicinal Chemistry;2024-05-09

3. Drug discovery targeting nicotinamide phosphoribosyltransferase (NAMPT): Updated progress and perspectives;Bioorganic & Medicinal Chemistry;2024-02

4. Recent advances of targeting nicotinamide phosphoribosyltransferase (NAMPT) for cancer drug discovery;European Journal of Medicinal Chemistry;2023-10

5. Melanoma and subcutaneous adipose tissue: Role of peritumoral adipokines in disease characterization and prognosis;Pigment Cell & Melanoma Research;2023-06-19