Structure based design of nicotinamide phosphoribosyltransferase (NAMPT) inhibitors from a phenotypic screen-Reference-Cited by-同舟云学术

Structure based design of nicotinamide phosphoribosyltransferase (NAMPT) inhibitors from a phenotypic screen

Published:2018-02 Issue:3 Volume:28 Page:365-370
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Palacios Daniel S.,Meredith Erik,Kawanami Toshio,Adams Christopher,Chen Xin,Darsigny Veronique,Geno Erin,Palermo Mark,Baird Daniel,Boynton Geoffrey,Busby Scott A.,George Elizabeth L.,Guy Chantale,Hewett Jeffrey,Tierney Laryssa,Thigale Sachin,Weihofen Wilhelm,Wang Louis,White Nicole,Yin Ming,Argikar Upendra A.

Funder

Novartis Institutes for Biomedical Research

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference23 articles.

1. NAD+ Metabolism and the Control of Energy Homeostasis: A Balancing Act between Mitochondria and the Nucleus

2. The NAD Biosynthesis Pathway Mediated by Nicotinamide Phosphoribosyltransferase Regulates Sir2 Activity in Mammalian Cells

3. NAMPT overexpression in prostate cancer and its contribution to tumor cell survival and stress response

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