A new method for filtering of reactive “warheads” of transition-state analog protease inhibitors
Author:
Publisher
Elsevier BV
Subject
Organic Chemistry,Drug Discovery,Pharmacology,General Medicine
Reference30 articles.
1. The resurgence of covalent drugs;Singh;Nature Reviews Drug Discovery,2011
2. Reversible covalent inhibition of a protein target;Lee;Angewantde Chemie International Edition,2012
3. Mechanistic basis of enzyme-targeted drugs;Robertson;Biochemistry,2005
4. The pharmacological landscape and therapeutic potential of serine hydrolases;Bachovchin;Nature Reviews Drug Discovery,2012
5. Covalent modifiers: an orthogonal approach to drug design;Potashman;Journal of Medicinal Chemistry,2009
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4. From Catalytic Mechanism to Rational Design of Reversible Covalent Inhibitors of Serine and Cysteine Hydrolases;Israel Journal of Chemistry;2014-05-12
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